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Letrozole: Is it Recommended for Bodybuilding?

by WikiStero.com

Letrozole is also known as Ferama or Letromina. It is originally developed to treat early breast cancer during the postmenopausal in women. It is also prescribed medication to treat breast cancer who already have received standard treatment with tamoxifen citrate for five years. Sometimes it is also used for advanced breast cancer treatment.

In this article, I will discuss the complete details of Letrozole for bodybuilding. Letrozole or Ferama is a nonsteroidal drug that is considered a reversible aromatase inhibitor. It is one potent and popular aromatase inhibitor drug that is often used to control the estrogenic side effects of steroids.

Most steroid users use this drug while performing aromatase steroid cycles like Dianabol and Testosterone. This drug can reduce water retention, gynecomastia issues, and high blood pressure during the cycles. Before moving forward, let’s get a quick look at its basic summary.


I. Letrozole Summary

This drug is originally developed to treat breast cancer in postmenopausal women. When it comes to bodybuilding use, it is one of the most popular aromatase inhibitor drugs, which is often used along with anabolic steroids. It is a powerful drug that has the ability to block estrogen levels in the body. The AI appeals to combat adverse estrogenic side effects of aromatase anabolic steroids.

It can lower the overall estrogen level in the body because it can block aromatase enzymes. Other popular SERMs drugs also control estrogen levels, but they only target very specific areas in the body. So, Letrozole is very effective in combating a wider range of estrogenic side effects which occur due to anabolic steroids. Mainly gynecomastia and water retention effects.

It can prevent the high blood pressure effects which come along when you face excess water retention. It is a helpful medication, so you can buy Letrozole online or over the counter with a prescription.



II. Working Of Letrozole

This drug directly acts to stop estrogen stimulation. This drug is also used to fight against infertility and as an anti-estrogen drug by steroid users. When it comes to fertility treatment, Letrozole stimulates ovulation. It is often prescribed to females who have fertility issues and want to have children. According to a clinical study, it is an effective and successful drug in treating fertility in women.

Professional sports players like bodybuilders or athletes who use aromatase anabolic steroids like testosterone or Dianabol often use Letrozole along with these drugs. The aim of using this drug is to build significant muscle mass quickly and also get lean muscles. Moreover, it can block the conversion of testosterone into estrogen, which allows steroid users to recover their testosterone levels.


III. What Are The Recommended Dose Of Letrozole?

People don’t require its higher dose because even at very low doses, potent Letrozole provides its full effects and positive effects. Unlike other SERMs or AIs, steroid users might take higher doses, but Letrozole is always used with lower doses, even if you use it as a medical treatment. Its higher dose is never recommended.

The recommended Letrozole dose during anabolic steroid use is between 0.5 mg to 1.25 mg every other day. A lower dose of 0.5 mg every other day is enough for the severe estrogenic side effects that male users face during the anabolic steroid cycle. You can increase the dose up to 1.25 mg to 2.5 mg per day for any severe gynecomastia symptoms. Make sure to take any expert advice before using a high dose.

For female users, it is advisable to take 0.5 mg every other day to get effective results. However, Letrozole is not recommended as the first choice for females because it can significantly reduce estrogen levels in the body; hence it is widely used for medical purposes in female users.


IV. Is Letrozole Useful As a Performance-enhancement?

Letrozole is an effective drug often used by anabolic steroid users as an aromatase inhibitor that can prevent estrogen formation. It can help to mitigate severe estrogenic side effects caused by anabolic steroids. It can reduce the unwanted feminizing impacts of anabolic steroids.

It is not helpful for performance enhancement, but it can combat severe side effects such as gynecomastia (male breast enlargement), water retention, and bloating effects. In addition, this drug is also helpful in boosting testosterone levels by preventing its breakdown.


V. What Are The Benefits Of Using Letrozole?

Letrozole  is an effective drug for steroid users to reverse symptoms of gynecomastia. It is an attractive drug because it can block the conversion of testosterone into estrogen, which can boost testosterone levels and reduce estrogen levels. This positively prevents water retention and leads to hard and dry muscle tissues. It is the best for gynecomastia. The other benefits are:

  • Prevent estrogenic side effects
  • Eliminate gynecomastia or its symptoms at the initial stage of the cycle
  • Save muscle tissue after the cycle of the catabolic process
  • Breakdown after taking anabolic steroids
  • Shut down the process of gynecomastia
  • Prescribed anti-breast cancer medication



VI. What Are The Side Effects Of Using Letrozole?

The effects of this drug vary as individual experiences, which means some people do not face any single side effects, and some might face adverse side effects. The good news is that if you take Letrozole with a recommended and lower dose, you will avoid all the possible side effects of it. A lower dose does not cause any problems for you.

Usually, Letrozole AI side effects are similar to Arimidex drugs. You may face muscle or joint pain, acne, fatigue, diarrhea, chest pain, or constipation. All of these side effects mainly occur in those women who use this drug to treat breast cancer for a longer period of time.

Letrozole is a well-tolerated drug by male users when they take lower doses. Many male users don’t face any single side effects at all. But if they take an excessive dose, it will increase the risk of different potential side effects. Let’s take a closer look at the side effects of Letrozole:

  • Fatigue
  • Muscles, bones, and joint pain
  • Changes cholesterol level
  • Rebound of estrogen
  • Hot flashes
  • Dizziness
  • Blur vision
  • Night vision
  • Sleeping disorder
  • Swelling in hands, feet, and ankle
  • Appetite loss
  • Headache


VII. Letrozole Vs. Arimidex

Both of these drugs belong class to aromatase inhibitors. Letrozole is often used to reduce the risk of breast cancer in post-menopasual women and also increase the chance to ovulate. Arimidex is prescribed medication to treat post-meopasual breast cancer which works by reducing estrogen levels in the body.

Both of these drugs cause almost the same side effects such as Nausea, vomiting, headache, dizziness, fatigue and many more.

Letrozole is often used greater than anastrozole because it can suppress the estrogen level greatly in the body and stop breast tumors from growing.




Letrozole is a popular aromatase inhibitor that is often used during an aromatase steroid cycle. It can completely block the conversion of testosterone into estrogen and effectively reduce estrogen levels in the body. It can be helpful to combat potential side effects of anabolic steroids, such as gynecomastia, water retention, and bloating effects.

In addition, it is prescribed medication to treat early breast cancer symptoms in postmenopause women. It is not the first choice for female bodybuilders or athletes because it can greatly reduce their estrogen level, which causes numerous health issues in them.

It is advisable to take a very low dose of Letrozole even if you use this drug for medical treatment because higher doses increase the risk of numerous side effects of it. However, it is not necessary that all users will face all the possible side effects because it depends on individual tolerance levels.

To get high-quality products, you can find Letrozole for sale from the different top resellers.

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